CautionMarevan

Warfarin

Vitamin K antagonist

Teratogen — avoid 6–12/40. Used only for mechanical heart valves after careful counselling.

Oral

First-line for

  • Mechanical heart valve (specialist only)

Mechanism

Inhibits vitamin K epoxide reductase → ↓ functional factors II, VII, IX, X and proteins C/S. Crosses placenta freely.

Warfarin embryopathy — “FACES”

  • F — Facial dysmorphism (nasal hypoplasia)
  • A — Atrophy of optic nerve
  • C — Chondrodysplasia punctata
  • E — Epiphyseal stippling
  • S — Stunted growth

Dosing

Target INR
Depends on valve type
Switch
To LMWH 6–12/40 + from 36/40

Contraindications

  • AbsolutePregnancy 6–12/40 (teratogen)
  • AbsoluteActive bleeding

Side effects

  • Bleeding
  • Skin necrosis (early protein C drop)
  • Purple toe syndrome

Fetal & maternal notes

  • Teratogenic 6–12/40 — embryopathy 5%.
  • Fetal intracranial haemorrhage risk in T3.
  • Safe in breastfeeding (not in milk).

Key interactions

  • NSAIDs

    Avoid

    ↑ INR + bleeding

  • Antibiotics

    Caution

    Variable — recheck INR

  • Vitamin K

    Caution

    Antagonises

Clinical pearls

  • 💡 Counsel pre-conception: switch to LMWH before 6/40 if possible.
  • 💡 Reversal: vitamin K + PCC (Beriplex).

Content last reviewed: REPLACE_ME (e.g. 2026-07)

Spotted something out of date? See our disclaimer or use Report an Error above.

For educational use only

Not medical advice. Verify dosing against the BNF and your local trust guidelines before prescribing.